A cikin ƙusoshin da ba'a sani ba ko haɗuwar haɗuwa (microbes, fungi), magunguna tare da mafi yawan hanyoyin yin aiki suna da muhimmanci. 5-NOC wani wakili ne mai rikitarwa mai rikitarwa a kan yawancin microorganisms da aka sani. Yana da tasiri a kan wasu mycoses.
5-NOC - abun da ke ciki
Babban sashi na miyagun ƙwayoyi a tambaya shi ne nitroxoline. Yana da wata magungunan sinadarai masu sifofi daga 8-hydroxyquinoline, yana hana jigidar DNA daga sel kwayoyin halitta kuma ya hana haifuwa. Ƙananan matakan da aka haɗa a cikin tsarin 5-NOC-kwamfutar hannu sun haɗa da:
- lactose monohydrate;
- calcium hydrogen phosphate;
- masarar masara;
- Povidone K25;
- colloidal silicon dioxide;
- tsabtace talc;
- magnesium stearate;
- crospovidone.
Ana samar da kwayoyi a cikin harsashi mai kariya, wanda ya ƙunshi abubuwa masu zuwa:
- carmellose sodium;
- acacia danko;
- colloidal silicon dioxide;
- Povidone K25;
- titanium dioxide;
- masarar masara;
- sucrose;
- tsabtace talc;
- calcium carbonate;
- launin abinci - rawaya "Sunset Sunset" (E110) da quinoline (E104).
5-NOC - nuni
An yi amfani da miyagun ƙwayoyi don magance mummunar cututtuka ko raunin ciwo na tsarin urinary da haihuwa. Tablets 5-NOC suna da tasiri a kan waɗannan kungiyoyin microorganisms:
- Gram-tabbataccen mairobic da anaerobic;
- ƴan magunguna da anaerobic gram-negative;
- mycoplasma ;
- Alamar daji ;
- Trichomonas;
- Mycobacterium tarin fuka;
- dermatophytes;
- mold fungi;
- dan takarar;
- pathogens sa mai zurfi da mai tsanani mycoses.
5-NOC - alamomi don amfani:
- cystitis;
- pyelonephritis ;
- Alamar bayani;
- urethritis;
- ciwon ƙwayar cuta (adenoma, carcinoma) na prostate;
- prostatitis;
- ƙwayoyin ƙwayoyin cuta a cikin mafitsara ko filin mai fita.
An yi amfani da shirin da aka tsara don hana kamuwa da cuta a cikin waɗannan yanayi:
- lokacin aikawa;
- gano magudi;
- cystoscopy ;
- catheterization.
5-NOC - sakamako masu illa
Magungunan kwayar cutar mai tsanani zai iya haifar da halayen jiki na jiki daga kowane tsarin. Wannan yana nufin da wuya ya haifar da sakamakon illa. A cikin lokuta masu ban mamaki, shiri na 5-NOC ya sa:
- tachycardia;
- vomiting;
- anorexia;
- Nausea;
- hana hanta aiki;
- dizziness;
- Hanyar neuritis (tare da shigarwa mai tsawo);
- kariya;
- rashin daidaito;
- ciwon kai;
- polyneuropathy;
- thrombocytopenia;
- Ƙara yawan haɗarin uric acid;
- urticaria;
- itching na fata;
- ataxia;
- kamawa da fitsari a cikin launi mai launin fata.
5-NOC contraindications
Wannan kayan aiki ba'a bada shawara ga mutum rashin haƙuri ga kowane abu mai ladabi da aka jera a sama, ciki har da magunguna masu magunguna da harsashi. An yi amfani da miyagun ƙwayoyi 5-NOC a karkashin irin wannan yanayi:
- ciki;
- Kayan aiki;
- nono;
- raguwa mai tsanani na hanta ko koda tare da yardawar creatinine na kasa da 20 ml / min (wanda aka umarce shi da wuya, tare da taka tsantsan);
- shekaru har zuwa shekaru 3.
Yadda za a dauki nauyin 5-NOC?
Yankin yau da kullum na magani yana dogara da shekaru da kuma ciwon wasu cututtuka na kullum. Manya a rana yana buƙatar 400 Mg na miyagun ƙwayoyi 5-NOC - aikace-aikacen ya shafi ɗaukar wannan kashi, raba zuwa sau 4, 100 MG (2 allunan) kafin abinci. Tare da ciwon kwayar cutar mai tsanani, an ninka kashi biyu (800 MG). Yara fiye da shekaru 5 an umarce su magani na 200-400 na kowace rana 24, kuma yara 3-5 - shekaru 200. Jigilar farfadowa ba ta wuce 2-4 makonni, idan ya cancanta, maimaita shi.
Tare da isasshen koda da kuma rashin lafiya, an yi amfani da 5-NOC tare da matsananciyar hankali - alamu na amfani ba su haɗa da cututtuka ba, amma a cikin cututtuka masu tsanani, za'a iya tsara kwayoyin. A cikin waɗannan lokuta, ɗauki 1 kwamfutar hannu sau 4 a rana. Wajibi ne a kula da yawan koda da kuma hanta zuwa jiyya da kuma kula da matakin halayyar creatinine.
5-NOC - aikace-aikace na cystitis
Sashin maganin antimicrobial ya dace da kashi 400 na nitroxoline a kowace 24 hours. 5-NOC tare da shawarar cystitis yana da kyau na kwanaki 10-21. An ƙayyade ainihin lokaci na farfadowa ta hanyar likitancin likitancin da ke kan gwaje gwaje-gwajen gwaje-gwaje, da tsananin mummunan tsari, da kuma kasancewa daga illa daga jiyya. Wani lokaci ma dole ne a kara shi zuwa wata daya, musamman idan an haɗu da kamuwa da cuta ko sakandare.
5-NOC tare da pyelonephritis
Maganin da aka bayyana a cikin babban tsari yana buƙatar taƙaitaccen maganin kwayoyin cutar, 400 mg kowace rana don makon 2-2.5. A cikin yanayin ci gaba na pyelonephritis, likitan urologist ya yanke shawarar yadda za'a dauki 5-NOC. Akwai makircinsu na tsawon lokaci (magani 2-3 don kwanaki 14) da bambance-bambancen karatu tare da amfani da miyagun ƙwayoyi a cikin ƙananan sashi (100-200 MG).
Wani lokaci yana daukan mafi kyawun liyafar 5-NOC - alamomi don amfani sun hada da siffofin mai tsanani na pyelonephritis:
- xanthogranulomatous;
- purulent;
- bala'i.
5-NOC a cikin ciki
Cikin dukan lokacin gestation, tsarin urinary mata na da matukar damuwa kuma yana iya zama mai saukin kaiwa ga ƙullun ƙwayoyin cuta. Saboda wannan, mahaifiyar da ake sa ransu suna da sha'awar 5-NOC - zan iya sha shi a lokacin daukar ciki da kuma abin da aka yi. An haramta wannan kwayar cutar a cikin wannan halin, saboda zai iya rinjayar ci gaba ko kuma samuwar tayin.
5-NOC analogues
Lokacin da ba'a iya amfani da miyagun ƙwayoyi na antimicrobial gabatarwa ko kuma yana haifar da mummunar sakamako mai lalacewa ba, dole ne a soke shi. Hanyar da za a maye gurbin takaddun 5-NOC ta hanyar amfani da ma'anarta ko jinsi. Akwai alamun analogs guda biyu zuwa ga miyagun ƙwayoyi da aka kwatanta:
- Nitroxoline (Jamus, Rasha);
- Uroksolin (Ukraine).
Anyi amfani da kwayar cutar ta farko tare da maida hankali daban-daban na sashi mai aiki, wanda ya dace da farfadowa tare da mafi girma. Amfani na biyu shi ne kawai a cikin Allunan da abun ciki na sinadarai na 50 MG. Idan ba a yarda da nitroxoline ko kayan da aka samo shi ba, to lallai ya zama dole don amfani da kwayar halitta. Wannan miyagun ƙwayoyi yana da kusan halaye masu kama da 5-NOC - mahimman alamomi don amfani, aikin antibacterial da kuma kayan aiki, amma wani abu daban-daban. Ana amfani da magunguna masu kyau a cikin nau'i na bacteriophages:
- dysentery polyvalent;
- intesties;
- idan;
- staphylococcal;
- Magani;
- Klebsiella pneumonia;
- Pseudomonas (pseudomonas);
- kolik-proteyny;
- salmonella.
Sauran kwayoyin halitta tare da alamomi iri iri:
- Fosmicin;
- Ureacid;
- Fosmural;
- Bernie;
- Fosmicin;
- Monural;
- Phosphoral;
- Urophosfabol;
- Cystoral;
- Fayil;
- Urofoscin;
- Phosphocin;
- Espa-Focine.